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ID: ALA1133152

Journal: Bioorg Med Chem Lett

Title: Design and synthesis of mimics of S-adenosyl-L-homocysteine as potential inhibitors of erythromycin methyltransferases.

Authors: Hanessian S, Sgarbi PW.

Abstract: A series of indanotriazine C-ribosides were prepared as SAH mimics, and tested for their ability to inhibit erythromycin resistance methylases Erm AM and Erm C'. A carbocyclic analogue derived from quinic acid was also synthesized and tested.

CiteXplore: 10743942

DOI: 10.1016/s0960-894x(00)00021-4