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ID: ALA1133199

Journal: Bioorg Med Chem Lett

Title: Synthesis and uptake of nitric oxide-releasing drugs by the P2 nucleoside transporter in Trypanosoma equiperdum.

Authors: Soulère L, Hoffmann P, Bringaud F, Périé J.

Abstract: A series of S-nitrosothiols, structurally related to the NO*-donor S-nitroso-N-acetylpenicillamine, and of organic nitrate esters that contain amidine groups which specify a recognition via the trypanosomal purine transporter P2, were synthesized and tested for their ability to inhibit the uptake of [2-(3)H]adenosine on Trypanosoma equiperdum.

CiteXplore: 10890161

DOI: 10.1016/s0960-894x(00)00233-x