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ID: ALA1133404

Journal: Bioorg Med Chem Lett

Title: Synthesis and biological activities of NB-506 analogues modified at the glucose group.

Authors: Ohkubo M, Nishimura T, Kawamoto H, Nakano M, Honma T, Yoshinari T, Arakawa H, Suda H, Morishima H, Nishimura S.

Abstract: A new indolocarbazole compound, NB-506 (1), modified at the glucose group yielded a beta-D-glucopyranoside, J-107,088 (2), which showed potent anticancer activity. A beta-D-ribofuranoside, J-109,534 (3), was found to be 6 times more potent than J-107,088 at inhibiting topoisomerase I.

CiteXplore: 10743939

DOI: 10.1016/s0960-894x(00)00004-4