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ID: ALA1134870

Journal: Bioorg Med Chem Lett

Title: Design and synthesis of novel inhibitors of gelatinase B.

Authors: Wang X, Choe Y, Craik CS, Ellman JA.

Abstract: A new method was developed to identify nonpeptidic metalloproteinase inhibitors with novel zinc binding groups. Application of this method to matrix metalloproteinase-9 resulted in the identification of aminomethyl benzimidazole analogue 7a with an IC(50)=13 microM.

CiteXplore: 12127537

DOI: 10.1016/s0960-894x(02)00365-7