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ID: ALA1134984

Journal: Bioorg Med Chem Lett

Title: Anticancer activity for 4,4'-dihydroxybenzophenone-2,4-dinitrophenylhydrazone (A-007) analogues and their abilities to interact with lymphoendothelial cell surface markers.

Authors: Morgan LR, Jursic BS, Hooper CL, Neumann DM, Thangaraj K, LeBlanc B.

Abstract: The structure of the anticancer agent 4,4'-dihydroxybenzophenone-2,4-dinitrophenylhydrazone (A-007) has been modified through SAR and by incorporating barbituric acid, pyridine, quinoline, and alkylcarboxylic acids into A-007's moieties. Analogue anticancer activity and interacting with CD surface markers on a T-cell leukemia cell line were evaluated and the correlation between SAR and biological properties are discussed.

CiteXplore: 12419372

DOI: 10.1016/s0960-894x(02)00725-4