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ID: ALA1135148

Journal: Bioorg Med Chem Lett

Title: Synthesis and profile of SCH351591, a novel PDE4 inhibitor.

Authors: Billah M, Cooper N, Cuss F, Davenport RJ, Dyke HJ, Egan R, Ganguly A, Gowers L, Hannah DR, Haughan AF, Kendall HJ, Lowe C, Minnicozzi M, Montana JG, Naylor R, Oxford J, Peake JC, Piwinski JJ, Runcie KA, Sabin V, Sharpe A, Shih NY, Warneck JB.

Abstract: The syntheses and pharmacological profiles of some 2-trifluoromethyl-8-methoxyquinoline-5-carboxamides are described. SCH351591 is a potent selective inhibitor of phosphodiesterase type 4 (PDE4).

CiteXplore: 12039576

DOI: 10.1016/s0960-894x(02)00225-1