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ID: ALA1135307

Journal: Bioorg Med Chem Lett

Title: Novel diamide-based inhibitors of IMPDH.

Authors: Gu HH, Iwanowicz EJ, Guo J, Watterson SH, Shen Z, Pitts WJ, Dhar TG, Fleener CA, Rouleau K, Sherbina NZ, Witmer M, Tredup J, Hollenbaugh D.

Abstract: A series of novel amide-based small molecule inhibitors of inosine monophosphate dehydrogenase is described. The synthesis and the structure-activity relationships (SARs) derived from in vitro studies are presented.

CiteXplore: 11965381

DOI: 10.1016/s0960-894x(02)00132-4