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ID: ALA1135864

Journal: Bioorg Med Chem Lett

Title: Novel amide-based inhibitors of inosine 5'-monophosphate dehydrogenase.

Authors: Watterson SH, Liu C, Dhar TG, Gu HH, Pitts WJ, Barrish JC, Fleener CA, Rouleau K, Sherbina NZ, Hollenbaugh DL, Iwanowicz EJ.

Abstract: A series of novel amide-based small molecule inhibitors of inosine monophosphate dehydrogenase (IMPDH) was explored. The synthesis and the structure-activity relationships (SARs) derived from in vitro studies are described.

CiteXplore: 12270168

DOI: 10.1016/s0960-894x(02)00601-7