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ID: ALA1136036

Journal: Bioorg Med Chem Lett

Title: Targeting thrombin and factor VIIa: design, synthesis, and inhibitory activity of functionally relevant indolizidinones.

Authors: Hanessian S, Therrien E, Granberg K, Nilsson I.

Abstract: Guided by molecular modeling, docking experiments, and available X-ray crystal structure data on the serine protease Factor VIIa and thrombin, a series of indolizidinone derivatives was designed and synthesized having diverse functionality at the P1, P2, and P3 sites.

CiteXplore: 12270173

DOI: 10.1016/s0960-894x(02)00612-1