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ID: ALA1136063

Journal: Bioorg Med Chem Lett

Title: Oxal hydroxamic acid derivatives with inhibitory activity against matrix metalloproteinases.

Authors: Krumme D, Tschesche H.

Abstract: Several amines, amino acid derivatives and low molecular weight peptides containing an amide-bound oxal hydroxamic acid moiety have been synthesized and tested for their inhibitory effects towards native human gelatinase B (MMP-9) and the catalytic domains of the membrane type MT1-MMP (MMP-14) and of neutrophil collagenase (MMP-8). A number of these compounds exhibited considerable inhibitory activity against the tested metalloproteinases.

CiteXplore: 11958997

DOI: 10.1016/s0960-894x(02)00052-5