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ID: ALA1136137

Journal: Bioorg Med Chem Lett

Title: Ring substituted analogues of 5-aminomethyl-10,11-dihydro-dibenzo[a,d]cycloheptene (AMDH): potential modes of binding to the 5-HT(2A) receptor.

Authors: Peddi S, Roth BL, Glennon RA, Westkaemper RB.

Abstract: The synthesis and 5-HT(2A) receptor affinities of 2-substituted-5-aminomethyl-10,11-dihydrodibenzo[a,d]cycloheptene (AMDH) derivatives are described. Comparison of the effects of substitution on affinities allowed assignment of potential binding modes in comparison with DOB-like agonists/antagonists and 3-substituted 1-(aminomethyl)-9,10-dihydroanthracene structures.

CiteXplore: 12852967

DOI: 10.1016/s0960-894x(03)00504-3