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ID: ALA1136534

Journal: Bioorg Med Chem Lett

Title: Dihydroquinolines with amine-containing side chains as potent n-NOS inhibitors.

Authors: Jaroch S, Hölscher P, Rehwinkel H, Sülzle D, Burton G, Hillmann M, McDonald FM.

Abstract: Dihydroquinolines with aminoalkyl side chains have been synthesized and have been shown to be potent n-NOS inhibitors. A marked selectivity versus e-NOS of up to approximately 300-fold was observed, whereas i-NOS was moderately inhibited.

CiteXplore: 12781178

DOI: 10.1016/s0960-894x(03)00351-2