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Basic Information

ID: ALA1141948

Journal: Bioorg Med Chem Lett

Title: Selective and orally bioavailable phenylglycine tissue factor/factor VIIa inhibitors.

Authors: Zbinden KG, Obst-Sander U, Hilpert K, Kühne H, Banner DW, Böhm HJ, Stahl M, Ackermann J, Alig L, Weber L, Wessel HP, Riederer MA, Tschopp TB, Lavé T.

Abstract: We describe the structure-based design and synthesis of highly potent, orally bioavailable tissue factor/factor VIIa inhibitors which interfere with the coagulation cascade by selective inhibition of the extrinsic pathway.

CiteXplore: 16213138

DOI: 10.1016/j.bmcl.2005.04.079