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ID: ALA1142791

Journal: Bioorg Med Chem Lett

Title: Design, synthesis, and evaluation of 2-phenoxy-indan-1-one derivatives as acetylcholinesterase inhibitors.

Authors: Sheng R, Lin X, Li J, Jiang Y, Shang Z, Hu Y.

Abstract: A series of 2-phenoxy-indan-1-one derivatives have been designed, synthesized, and tested as acetylcholinesterase inhibitors. The most potent compound exhibited high AChE inhibitory activity (IC50 = 50 nM), and the molecular docking study indicated that it was nicely accommodated by AChE.

CiteXplore: 15993600

DOI: 10.1016/j.bmcl.2005.05.132