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ID: ALA1144791

Journal: Bioorg Med Chem Lett

Title: Facile synthesis of substituted trans-2-arylcyclopropylamine inhibitors of the human histone demethylase LSD1 and monoamine oxidases A and B.

Authors: Gooden DM, Schmidt DM, Pollock JA, Kabadi AM, McCafferty DG.

Abstract: A facile synthetic route to substituted trans-2-arylcyclopropylamines was developed to provide access to mechanism-based inhibitors of the human flavoenzyme oxidase lysine-specific histone demethylase LSD1 and related enzyme family members such as monoamine oxidases A and B.

CiteXplore: 18242989

DOI: 10.1016/j.bmcl.2008.01.003