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ID: ALA1144977

Journal: Bioorg Med Chem Lett

Title: Synthesis of pyrimidinopyridine-triazene conjugates targeted to abl tyrosine kinase.

Authors: Rachid Z, Katsoulas A, Brahimi F, Jean-Claude BJ.

Abstract: The synthesis and abl tyrosine kinase inhibitory activities of alkyltriazenes conjugated to phenylaminopyrimidines are described. Significant abl inhibitory activities were observed only when a benzamido spacer was inserted between the 1,2,3-triazene chain and the 2-phenyaminopyridopyrimidine moiety.

CiteXplore: 12951113

DOI: 10.1016/s0960-894x(03)00553-5