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ID: ALA1146650

Journal: Bioorg Med Chem Lett

Title: 1,7-annulated indolocarbazoles as cyclin-dependent kinase inhibitors.

Authors: Al-awar RS, Ray JE, Hecker KA, Huang J, Waid PP, Shih C, Brooks HB, Spencer CD, Watkins SA, Patel BR, Stamm NB, Ogg CA, Schultz RM, Considine EL, Faul MM, Sullivan KA, Kolis SP, Grutsch JL, Joseph S.

Abstract: The synthesis and kinase inhibitory activity of a series of novel 1,7-annulated indolocarbazoles 6 and 16 is described. These compounds exhibited potent inhibitory activity against cyclin-dependent kinase 4 and good antiproliferative activity in a human colon carcinoma cell line.

CiteXplore: 15149678

DOI: 10.1016/j.bmcl.2004.03.105