Document Report Card

Basic Information

ID: ALA1147640

Journal: Bioorg Med Chem Lett

Title: Antitumor agents. Part 232: Synthesis of cyclosulfite podophyllotoxin analogues as novel prototype antitumor agents.

Authors: Xiao Z, Han S, Bastow KF, Lee KH.

Abstract: An 11,13-O,O'-cyclosulfite GL-331 analogue (7) was synthesized in six steps from podophyllotoxin and evaluated as a potential antitumor agent. Compound 7 was significantly cytotoxic against human tumor cell lines, but showed no inhibition against human DNA topoisomerase II in vitro. This compound represents a novel prototype of antitumor podophyllotoxin analogues.

CiteXplore: 15006408

DOI: 10.1016/j.bmcl.2003.12.096