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ID: ALA1147762

Journal: Bioorg Med Chem Lett

Title: A new chemical tool for exploring the physiological function of the PDE2 isozyme.

Authors: Chambers RJ, Abrams K, Garceau NY, Kamath AV, Manley CM, Lilley SC, Otte DA, Scott DO, Sheils AL, Tess DA, Vellekoop AS, Zhang Y, Lam KT.

Abstract: Oxindole (2) is a potent and selective PDE2 inhibitor with a favorable ADME, physiochemical and pharmacokinetic profile to allow for use as a chemical tool in elucidating the physiological role of PDE2.

CiteXplore: 16275071

DOI: 10.1016/j.bmcl.2005.10.005