Document Report Card

Basic Information

ID: ALA1147773

Journal: Bioorg Med Chem Lett

Title: Potent anti-muscarinic activity in a novel series of quinuclidine derivatives.

Authors: Starck JP, Talaga P, Quéré L, Collart P, Christophe B, Lo Brutto P, Jadot S, Chimmanamada D, Zanda M, Wagner A, Mioskowski C, Massingham R, Guyaux M.

Abstract: The synthesis and biological evaluation of a novel family of M(3) muscarinic antagonists are described. A systematic modification of the substituents to a novel alkyne-quinuclidine scaffold yielded original compounds displaying potent in vitro anticholinergic properties.

CiteXplore: 16275087

DOI: 10.1016/j.bmcl.2005.09.079