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ID: ALA1151865

Journal: Bioorg Med Chem Lett

Title: New developments for the design, synthesis and biological evaluation of potent SARS-CoV 3CL(pro) inhibitors.

Authors: Regnier T, Sarma D, Hidaka K, Bacha U, Freire E, Hayashi Y, Kiso Y.

Abstract: A series of trifluoromethyl, benzothiazolyl or thiazolyl ketone-containing peptidic compounds as SARS-CoV 3CL protease inhibitors were developed and their potency was evaluated by in vitro protease inhibitory assays. Three candidates had encouraging results for the development of new anti-SARS compounds.

CiteXplore: 19362479

DOI: 10.1016/j.bmcl.2009.03.118