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ID: ALA1153266

Journal: Bioorg Med Chem Lett

Title: Synthesis and biological activity of anticoccidial agents: 2,3-diarylindoles.

Authors: Scribner A, Moore JA, Ouvry G, Fisher M, Wyvratt M, Leavitt P, Liberator P, Gurnett A, Brown C, Mathew J, Thompson D, Schmatz D, Biftu T.

Abstract: Novel 2,3-diarylindoles bearing an amine substituent at the indole 5- and 6-positions have been synthesized and evaluated as anticoccidial agents in both in vitro and in vivo assays. Both subnanomolar in vitro activity and broad spectrum in vivo potency were detected for several compounds, particularly compound 27.

CiteXplore: 19195883

DOI: 10.1016/j.bmcl.2009.01.001