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ID: ALA1177821

Journal: Bioorg Med Chem Lett

Title: Structure-activity relationships and hepatic safety risks of thiazole agonists of the thrombopoietin receptor.

Authors: Antipas AS, Blumberg LC, Brissette WH, Brown MF, Casavant JM, Doty JL, Driscoll J, Harris TM, Jones CS, McCurdy SP, McElroy E, Mitton-Fry M, Munchhof MJ, Reim DA, Reiter LA, Ripp SL, Shavnya A, Smeets MI, Trevena KA.

Abstract: 5-F substitution of an aminothiazole moiety within a series of thrombopoietin receptor agonists leads to potent agents with an improved hepatic safety profile in rodent toxicology studies.

CiteXplore: 20558059

DOI: 10.1016/j.bmcl.2010.05.087