Document Report Card

Basic Information

ID: ALA1828604

Journal: Bioorg Med Chem

Title: Antifungal activity of a series of 1,2-benzisothiazol-3(2H)-one derivatives.

Authors: Dou D, Alex D, Du B, Tiew KC, Aravapalli S, Mandadapu SR, Calderone R, Groutas WC.

Abstract: A series of broad-spectrum antifungal agents based on the 1,2-benzisothiazol-3(2H)-one scaffold is reported. Preliminary structure-activity relationship studies have established the importance of the presence of the heterocyclic ring, a methyl group, and a phenyl ring for optimal manifestation of antifungal activity.

CiteXplore: 21903403

DOI: 10.1016/j.bmc.2011.08.029