Document Report Card

Basic Information

ID: ALA1909601

Journal: Bioorg Med Chem Lett

Title: Synthesis and structure-activity relationship studies of dihydronaphthyridinediones as a novel structural class of potent and selective PDE7 inhibitors.

Authors: Gewald R, Rueger C, Grunwald C, Egerland U, Hoefgen N.

Abstract: The synthesis and SAR studies of a series of structurally novel inhibitors of PDE7 are discussed. The best compounds from the series display low nanomolar inhibitory activity and are selective versus other PDE isoenzymes.

CiteXplore: 21983442

DOI: 10.1016/j.bmcl.2011.09.065