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ID: ALA1914314

Journal: Bioorg Med Chem Lett

Title: Acidic triazoles as soluble guanylate cyclase stimulators.

Authors: Roberts LR, Bradley PA, Bunnage ME, England KS, Fairman D, Fobian YM, Fox DN, Gymer GE, Heasley SE, Molette J, Smith GL, Schmidt MA, Tones MA, Dack KN.

Abstract: A series of acidic triazoles with activity as soluble guanylate cyclase stimulators is described. Incorporation of the CF(3) triazole improved the overall physicochemical and drug-like properties of the molecule and is exemplified by compound 25.

CiteXplore: 21924901

DOI: 10.1016/j.bmcl.2011.08.071