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Basic Information

ID: ALA1955823

Journal: Bioorg Med Chem Lett

Title: Imidazo[1,2-a]pyrazines as novel PI3K inhibitors.

Authors: Martínez González S, Hernández AI, Varela C, Rodríguez-Arístegui S, Alvarez RM, García AB, Lorenzo M, Rivero V, Oyarzabal J, Rabal O, Bischoff JR, Albarrán M, Cebriá A, Alfonso P, Link W, Fominaya J, Pastor J.

Abstract: Phosphoinositide-3-kinase (PI3K) is an important target for cancer therapeutics due to the deregulation of its signaling pathway in a wide variety of human cancers. We describe herein a novel series of imidazo[1,2-a]pyrazines as PI3K inhibitors.

CiteXplore: 22325943

DOI: 10.1016/j.bmcl.2012.01.074