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ID: ALA2434955

Journal: Bioorg Med Chem Lett

Title: Potent inhibition of norovirus by dipeptidyl α-hydroxyphosphonate transition state mimics.

Authors: Mandadapu SR, Gunnam MR, Galasiti Kankanamalage AC, Uy RA, Alliston KR, Lushington GH, Kim Y, Chang KO, Groutas WC.

Abstract: The design, synthesis, and evaluation of a series of dipeptidyl α-hydroxyphosphonates is reported. The synthesized compounds displayed high anti-norovirus activity in a cell-based replicon system, as well as high enzyme selectivity.

CiteXplore: 24054123

DOI: 10.1016/j.bmcl.2013.08.073