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ID: ALA3286210

Journal: Bioorg Med Chem Lett

Title: Discovery of 3-aryl-3-ethoxypropanoic acids as orally active GPR40 agonists.

Authors: Takano R, Yoshida M, Inoue M, Honda T, Nakashima R, Matsumoto K, Yano T, Ogata T, Watanabe N, Toda N.

Abstract: The G protein-coupled receptor 40 (GPR40) mediates enhancement of glucose-stimulated insulin secretion in pancreatic β cells. The GPR40 agonist has been attracting attention as a novel insulin secretagogue with glucose dependency for the treatment of type 2 diabetes. The optimization study of compound 1 led to a potent and bioavailable GPR40 agonist 24, which showed insulin secretion and glucose lowering effects in rat OGTT. Compound 24 is a potential lead compound for a novel insulin secretagogue with a low risk of hypoglycemia.

CiteXplore: 24835985

DOI: 10.1016/j.bmcl.2014.04.065