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ID: ALA3603743

Journal: Bioorg Med Chem

Title: Design, synthesis and biological evaluation of saccharin-based N-hydroxybenzamides as histone deacetylases (HDACs) inhibitors.

Authors: Fu H, Han L, Hou X, Dun Y, Wang L, Gong X, Fang H.

Abstract: We report the development of a novel series of saccharin-based N-hydroxybenzamides as histone deacetylases inhibitors. Among them, 6 j exhibited potent HDACs inhibitory activity against Hela nuclear extract. Further biological evaluation found 6 i showed similar antiproliferative activities in vitro compared with the approved SAHA.

CiteXplore: 26216016

DOI: 10.1016/j.bmc.2015.07.008