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ID: ALA4425182

Journal: Bioorg Med Chem Lett

Title: Trypsin inhibitors for the treatment of pancreatitis.

Authors: Brandl T, Simic O, Skaanderup PR, Namoto K, Berst F, Ehrhardt C, Schiering N, Mueller I, Woelcke J.

Abstract: Proline-based trypsin inhibitors occupying the S1-S2-S1' region were identified by an HTS screening campaign. It was discovered that truncation of the P1' moiety and appropriate extension into the S4 region led to highly potent trypsin inhibitors with excellent selectivity against related serine proteases and a favorable hERG profile.

CiteXplore: 27476144

DOI: 10.1016/j.bmcl.2016.07.029