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ID: ALA4507296
Title: Data for DCP probe PF-05105679
Authors: SGC Frankfurt
Abstract: SGC Frankfurt donated chemical probe project: PF-05105679 was donated by Pfizer. Website: https://www.sgc-ffm.uni-frankfurt.de/#!specificprobeoverview/PF-05105679. Control: PF-05257137. References: 1. Andrews, Mark D, Kerry Af Forselles, Kevin Beaumont, Sébastien R G Galan, Paul A Glossop, Mathilde Grenie, Alan Jessiman, Amy S Kenyon, Graham Lunn, Graham Maw, Robert M Owen, David C Pryde, Dannielle Roberts, and Thien Duc Tran. 2015. ‘Discovery of a Selective TRPM8 Antagonist with Clinical Efficacy in Cold-Related Pain’. ACS Medicinal Chemistry Letters 6(4):419–24. PMID: 25893043. 2. Winchester, Wendy J, Katrina Gore, Sophie Glatt, Wendy Petit, Jennifer C Gardiner, Kelly Conlon, Michael Postlethwaite, Pierre-Philippe Saintot, Sonia Roberts, James R Gosset, Tomomi Matsuura, Mark D Andrews, Paul A Glossop, Michael J Palmer, Nicola Clear, Susie Collins, Kevin Beaumont, and David S Reynolds. 2014. ‘Inhibition of TRPM8 Channels Reduces Pain in the Cold Pressor Test in Humans’. The Journal of Pharmacology and Experimental Therapeutics 351(2):259–69. PMID: 25125580.