Data for DCP probe (R)-9s

Basic Information

ID: ALA4507301

Title: Data for DCP probe (R)-9s

Authors: SGC Frankfurt

Abstract: SGC Frankfurt donated chemical probe project: (R)-9s was donated by Takeda. Website: https://www.sgc-ffm.uni-frankfurt.de/#!specificprobeoverview/(R)-9s. Control: (S)-9s. References: 1. Sakauchi, Nobuki, Yasuhisa Kohara, Ayumu Sato, Tomohiko Suzaki, Yumi Imai, Yuichi Okabe, Shigemitsu Imai, Reiko Saikawa, Hiroshi Nagabukuro, Haruhiko Kuno, Hisashi Fujita, Izumi Kamo, and Masato Yoshida. 2016. ‘Discovery of 5-Chloro-1-(5-Chloro-2-(Methylsulfonyl)Benzyl)-2-Imino-1,2-Dihydropyridine-3-Carboxamide (TAK-259) as a Novel, Selective, and Orally Active Α1D Adrenoceptor Antagonist with Antiurinary Frequency Effects: Reducing Human Ether-a-Go-Go-Related Gene (HERG) Liabilities’. Journal of Medicinal Chemistry 59(7):2989–3002. PMID: 26954848.

DOI: 10.6019/CHEMBL4507301

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