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Bradykinin B1 receptor

Name And Classification

ID:  ALA4613

Type:  SINGLE PROTEIN

Synonyms:   B1 bradykinin receptor | B1bkr | B1R | Bdkrb1 | BK-1 receptor | Bkr | KB1 | Kinin B1 receptor

Organism:  Rattus norvegicus

Species Group:  Rattus norvegicus

Protein Target Classification:   Membrane receptor / Family A G protein-coupled receptor / Peptide receptor (family A GPCR) / Short peptide receptor (family A GPCR) / Bradykinin receptor

Target Components

DescriptionRelationshipAccession
B1 bradykinin receptorPROTEINP97583

Associated Recombinant Proteins

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NameSpecification and purityExpression systemProtein labelActivityView Details

Associated Active Ligands

  1. Tetrahydrouridine
    ALA299832

    Name:
    1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-(4-(4-(pyridin-4-yl)piperazin-1-yl)phenyl)urea

    Mol. Formula:
    C36H39N7O2

    M.W.:
    601.76

    Type:
    Small molecule

    AlogP:
    5.73

    Polar Surface Area:
    93.17

    HBA:
    6

    HBD:
    2

    #RO5 Violations:
    2

    #Rotatable Bonds:
    9

    Passes Ro3:
    N

    QED Weighted:
    0.26

    DETAILS
  2. Tetrahydrouridine
    ALA315388

    Name:
    (S)-2-{[(S)-1-((S)-2-{13-[(S)-2-((S)-2,6-Diamino-hexanoylamino)-5-guanidino-pentanoylamino]-tridecanoylamino}-3-hydroxy-propionyl)-pyrrolidine-2-carbonyl]-amino}-3-phenyl-propionic acid

    Mol. Formula:
    C42H72N10O8

    M.W.:
    845.10

    Type:
    Small molecule

    AlogP:
    0.67

    Polar Surface Area:
    310.68

    HBA:
    10

    HBD:
    10

    #RO5 Violations:
    2

    #Rotatable Bonds:
    32

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS
  3. Tetrahydrouridine
    ALA406554

    Name:
    H-Lys-Arg-Gly-Gly-Gly-Ser-Pro-Phe-OH

    Mol. Formula:
    C35H56N12O10

    M.W.:
    804.91

    Type:
    Protein

    AlogP:
    -5.39

    Polar Surface Area:
    368.88

    HBA:
    12

    HBD:
    12

    #RO5 Violations:
    3

    #Rotatable Bonds:
    25

    Passes Ro3:
    N

    QED Weighted:
    0.02

    DETAILS
  4. Tetrahydrouridine
    ALA431264

    Name:
    H-Lys-Arg-Gly-1-amino-1-carboxycyclododecane-Gly-Ser-Pro-Phe-OH

    Mol. Formula:
    C46H76N12O10

    M.W.:
    957.19

    Type:
    Protein

    AlogP:
    -1.35

    Polar Surface Area:
    368.88

    HBA:
    12

    HBD:
    12

    #RO5 Violations:
    3

    #Rotatable Bonds:
    25

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS
  5. Tetrahydrouridine
    ALA329578

    Name:
    H-Lys-Arg-Gly-1-amino-1-carboxycyclononane-Gly-Ser-Pro-Phe-OH

    Mol. Formula:
    C43H70N12O10

    M.W.:
    915.11

    Type:
    Protein

    AlogP:
    -2.52

    Polar Surface Area:
    368.88

    HBA:
    12

    HBD:
    12

    #RO5 Violations:
    3

    #Rotatable Bonds:
    25

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS
  6. Tetrahydrouridine
    ALA96398

    Name:
    H-Lys-Arg-1-amino-1-carboxycycloheptane-Ser-Pro-Phe-OH

    Mol. Formula:
    C37H60N10O8

    M.W.:
    772.95

    Type:
    Protein

    AlogP:
    -1.53

    Polar Surface Area:
    310.68

    HBA:
    10

    HBD:
    10

    #RO5 Violations:
    2

    #Rotatable Bonds:
    21

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS
  7. Tetrahydrouridine
    ALA96119

    Name:
    H-Lys-Arg-Gly-1-amino-1-carboxycyclooctane-Gly-Ser-Pro-Phe-OH

    Mol. Formula:
    C42H68N12O10

    M.W.:
    901.08

    Type:
    Protein

    AlogP:
    -2.91

    Polar Surface Area:
    368.88

    HBA:
    12

    HBD:
    12

    #RO5 Violations:
    3

    #Rotatable Bonds:
    25

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS
  8. Tetrahydrouridine
    ALA313869

    Name:
    H-Lys-Arg-Gly-1-amino-1-carboxycycloheptane-Gly-Ser-Pro-Phe-OH

    Mol. Formula:
    C41H66N12O10

    M.W.:
    887.05

    Type:
    Protein

    AlogP:
    -3.30

    Polar Surface Area:
    368.88

    HBA:
    12

    HBD:
    12

    #RO5 Violations:
    3

    #Rotatable Bonds:
    25

    Passes Ro3:
    N

    QED Weighted:
    0.02

    DETAILS
  9. Tetrahydrouridine
    ALA318524

    Name:
    H-Lys-Arg-Gly-1-amino-1-carboxycyclohexane-Gly-Ser-Pro-Phe-OH

    Mol. Formula:
    C40H64N12O10

    M.W.:
    873.03

    Type:
    Protein

    AlogP:
    -3.69

    Polar Surface Area:
    368.88

    HBA:
    12

    HBD:
    12

    #RO5 Violations:
    3

    #Rotatable Bonds:
    25

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS
  10. Tetrahydrouridine
    ALA320458

    Name:
    Lys-Arg-4-aminododecanoic acid-Ser-Pro-Phe

    Mol. Formula:
    C41H70N10O8

    M.W.:
    831.07

    Type:
    Small molecule

    AlogP:
    0.28

    Polar Surface Area:
    310.68

    HBA:
    10

    HBD:
    10

    #RO5 Violations:
    2

    #Rotatable Bonds:
    31

    Passes Ro3:
    N

    QED Weighted:
    0.03

    DETAILS