# | Name | Compound Key | Action Type | Relation | Activety Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | [³H]melatonin | 1 | Ki | = | 0.429 | nM | ALA2328137 | 9.37 | nM | Homo sapiens | ||
2. | ALA2326199 | 1 | Ki | = | 0.291 | nM | ALA2328137 | 9.54 | nM | Homo sapiens | ||
3. | ALA2326200 | 7 | Ki | = | 0.073 | nM | ALA2328137 | 10.14 | nM | Homo sapiens | ||
4. | ALA2326201 | 8 | Ki | = | 0.55 | nM | ALA2328137 | 9.26 | nM | Homo sapiens | ||
5. | BOMPPA | 9 | Ki | = | 3.39 | nM | ALA2328137 | 8.47 | nM | Homo sapiens | ||
6. | ALA2326203 | 10 | Ki | = | 0.339 | nM | ALA2328137 | 9.47 | nM | Homo sapiens | ||
7. | ALA2326199 | 1 | EC50 | = | 0.05 | nM | ALA2328004 | 10.30 | nM | Homo sapiens | ||
8. | ALA2326200 | 7 | EC50 | = | 0.11 | nM | ALA2328004 | 9.96 | nM | Homo sapiens | ||
9. | ALA2326201 | 8 | EC50 | = | 0.024 | nM | ALA2328004 | 10.62 | nM | Homo sapiens | ||
10. | BOMPPA | 9 | EC50 | = | 0.24 | nM | ALA2328004 | 9.62 | nM | Homo sapiens | ||
11. | ALA2326203 | 10 | EC50 | = | 0.2 | nM | ALA2328004 | 9.70 | nM | Homo sapiens | ||
12. | ALA2314255 | 9e | Ki | = | 0.03 | nM | ALA2318043 | 10.52 | nM | Homo sapiens | ||
13. | 2-methoxy-α,β-didehydro-agomelatine | 9g | Ki | = | 0.07 | nM | ALA2318043 | 10.15 | nM | Homo sapiens | ||
14. | ALA2314257 | 9f | Ki | = | 0.09 | nM | ALA2318043 | 10.05 | nM | Homo sapiens | ||
15. | Agomelatine | 1 | Ki | = | 0.1 | nM | ALA2318043 | 10.00 | nM | Homo sapiens | ||
16. | ALA2314253 | (+/-)-trans-8g | Ki | = | 0.2 | nM | ALA2318043 | 9.70 | nM | Homo sapiens | ||
17. | ALA2314260 | 10g | Ki | = | 0.3 | nM | ALA2318043 | 9.52 | nM | Homo sapiens | ||
18. | [³H]melatonin | 1 | Ki | = | 0.5 | nM | ALA2318043 | 9.30 | nM | Homo sapiens | ||
19. | ALA2314251 | (+/-)-trans-8e | Ki | = | 0.7 | nM | ALA2318043 | 9.15 | nM | Homo sapiens | ||
20. | ALA229015 | 4t | Ki | = | 1.4 | nM | ALA2318043 | 8.85 | nM | Homo sapiens |