# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | [³H]rolipram | 1 | IC50 | = | 0.5 | uM | ALA5237521 | 6.30 | nM | Homo sapiens | ||
2. | ALA5275470 | 44 | EC50 | = | 0.3 | uM | ALA5236710 | 6.52 | nM | Homo sapiens | ||
3. | ALA478482 | C35 | IC50 | = | 20.57 | uM | ALA5231474 | 4.69 | nM | Homo sapiens | ||
4. | ALA5282465 | 52 | IC50 | = | 0.89 | uM | ALA5231474 | 6.05 | nM | Homo sapiens | ||
5. | ALA5289737 | 51 | IC50 | = | 1.16 | uM | ALA5231474 | 5.94 | nM | Homo sapiens | ||
6. | ALA2391027 | 12d | IC50 | = | 3.31 | uM | ALA5231474 | 5.48 | nM | Homo sapiens | ||
7. | ALA5287859 | 40 | IC50 | = | 6.38 | uM | ALA5231474 | 5.20 | nM | Homo sapiens | ||
8. | ALA5268975 | 7 | IC50 | = | 0.629 | uM | ALA5231474 | 6.20 | nM | Homo sapiens | ||
9. | ALA5285518 | 6 | IC50 | = | 1.424 | uM | ALA5231474 | 5.85 | nM | Homo sapiens | ||
10. | UCB-9260 | 1a | Kd | = | 13 | nM | ALA5228021 | 7.89 | nM | Homo sapiens | ||
11. | ALA5270115 | 4; SPD-304 | Kd | = | 91.7 | uM | ALA5228020 | 4.04 | nM | Homo sapiens | ||
12. | ALA4457006 | 34 | Kd | = | 93.6 | uM | ALA4397827 | 4.03 | nM | Homo sapiens | ||
13. | ALA4793924 | 12 | t1/2 | = | 0.9 | hr | ALA4775693 | hr | Homo sapiens | |||
14. | ALA4787790 | 11 | t1/2 | = | 62.3 | hr | ALA4775693 | hr | Homo sapiens | |||
15. | ALA4793441 | 10 | t1/2 | = | 42.8 | hr | ALA4775693 | hr | Homo sapiens | |||
16. | ALA4793924 | 12 | IC50 | = | 71 | nM | ALA4775692 | 7.15 | nM | Homo sapiens | ||
17. | ALA4787790 | 11 | IC50 | = | 163 | nM | ALA4775692 | 6.79 | nM | Homo sapiens | ||
18. | ALA4793441 | 10 | IC50 | = | 189 | nM | ALA4775692 | 6.72 | nM | Homo sapiens | ||
19. | ALA4779860 | 9 | IC50 | = | 5300 | nM | ALA4775692 | 5.28 | nM | Homo sapiens | ||
20. | ALA1507048 | SID47204099 | IC50 | 0 | ALA4775692 | Not Determined | Homo sapiens |