# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BFH772 | 1 | IC50 | > | 0.5 | uM | ALA5252781 | nM | Homo sapiens | |||
2. | BAW2881(NVP-BAW2881) | 2 | IC50 | > | 0.5 | uM | ALA5252781 | nM | Homo sapiens | |||
3. | ALA5284848 | 14d | Activity | 0 | ALA5250208 | Active | Homo sapiens | |||||
4. | ALA4575427 | Tauroacidin B | IC50 | = | 37.93 | uM | ALA5243758 | 4.42 | nM | Homo sapiens | ||
5. | ALA1095259 | tauroacidin A | IC50 | = | 37.93 | uM | ALA5243758 | 4.42 | nM | Homo sapiens | ||
6. | ALA4539558 | Spongiacidin B | IC50 | = | 18.46 | uM | ALA5243758 | 4.73 | nM | Homo sapiens | ||
7. | ALA4531006 | Spongiacidin A | IC50 | = | 20.99 | uM | ALA5243758 | 4.68 | nM | Homo sapiens | ||
8. | ALA5286014 | 10; TAS0728 | IC50 | = | 13 | nM | ALA5243470 | 7.89 | nM | Homo sapiens | ||
9. | mobocertinib | MOBOCERTINIB | INH | > | 97 | % | ALA5238870 | % | Homo sapiens | |||
10. | Neratinib (HKI-272) | 25o (table 3) | IC50 | = | 59 | nM | ALA5233314 | 7.23 | nM | Homo sapiens | ||
11. | ALA5285419 | DTPA-A9 | Kd | = | 103 | nM | ALA5231951 | 6.99 | nM | Homo sapiens | ||
12. | ALA5285419 | DTPA-A9 | Kd | = | 4.9 | nM | ALA5231950 | 8.31 | nM | Homo sapiens | ||
13. | ALA5286730 | 33 | IC50 | = | 5.4 | uM | ALA5230878 | 5.27 | nM | Homo sapiens | ||
14. | Gefitinib (ZD1839) | Iressa | IC50 | = | 9.42 | uM | ALA5230878 | 5.03 | nM | Homo sapiens | ||
15. | MnTMPyP pentachloride | 5 | IC50 | = | 0.13 | uM | ALA5230847 | 6.89 | nM | Homo sapiens | ||
16. | ALA5199520 | 53j | IC50 | = | 0.17 | uM | ALA5230847 | 6.77 | nM | Homo sapiens | ||
17. | ALA5270336 | 13 | IC50 | = | 1.32 | uM | ALA5230836 | 5.88 | nM | Homo sapiens | ||
18. | Erlotinib | Tarceva | IC50 | = | 1.23 | uM | ALA5230836 | 5.91 | nM | Homo sapiens | ||
19. | ALA5281270 | 12c | IC50 | = | 0.042 | uM | ALA5230832 | 7.38 | nM | Homo sapiens | ||
20. | ALA5280584 | 12b | IC50 | = | 0.021 | uM | ALA5230832 | 7.68 | nM | Homo sapiens |