Activities

JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

The page will load shortly, Thanks for your patience!

྾

Activities

Select ☑️ to add compounds to your custom library, then export your list as CSV / TSV. See how it works.

#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA1614701	AZD-6244	AC50	>	10	uM	ALA5291809		Summarised AC50 (mean value for measurements with a relation sign "="; largest value for measurements with relation sign ">")	nM	Homo sapiens
2.	ALA1614701	AZD-6244	IC50	=	14	nM	ALA3751471	7.85		nM	Homo sapiens
3.	ALA1614701	AZD-6244	IC50	=	3.7	uM	ALA3751470	5.43		nM	Homo sapiens
4.	ALA1614701	AZD-6244	t1/2	=	4.1	hr	ALA3750101			hr	Rattus norvegicus
5.	ALA1614701	AZD-6244	IC50	>	10000	nM	ALA3751464			nM	Homo sapiens
6.	ALA1614701	AZD-6244	IC50	=	1750	nM	ALA3751463	5.76		nM	Homo sapiens
7.	ALA1614701	AZD-6244	IC50	=	69	nM	ALA3751462	7.16		nM
8.	ALA1614701	AZD-6244	IC50	=	32	nM	ALA3751461	7.50		nM	Homo sapiens
9.	ALA1614701	AZD-6244	BPR	<	0.02		ALA3751460
10.	ALA1614701	AZD-6244	F	=	24	%	ALA3751459			%	Rattus norvegicus
11.	ALA1614701	AZD-6244	Vdss	=	0.2	L/Kg	ALA3750098			L.kg-1	Rattus norvegicus
12.	ALA1614701	AZD-6244	CL	=	0.06	L/kg/hr	ALA3750095			mL.min-1.kg-1	Rattus norvegicus
13.	ALA1614701	AZD-6244	IC50	=	3000	nM	ALA3750090	5.52		nM
14.	ALA1614701	AZD-6244	IC50	=	31	nM	ALA3750088	7.51		nM	Homo sapiens
15.	ALA1614701	AZD-6244	IC50	=	0.95	uM	ALA5226853	6.02		nM	Homo sapiens
16.	ALA1614701	AZD-6244	IC50	=	1.25	uM	ALA5226852	5.90		nM	Homo sapiens
17.	ALA1614701	AZD-6244	Kd	=	530	nM	ALA5213094	6.28		nM	Homo sapiens
18.	ALA1614701	AZD-6244	Kd	=	99	nM	ALA5213093	7.00		nM	Homo sapiens
19.	ALA1614701	AZD-6244	Kd	=	530	nM	ALA5210362	6.28		nM	Homo sapiens
20.	ALA1614701	AZD-6244	Kd	=	99	nM	ALA5210361	7.00		nM	Homo sapiens