# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1630575 | caspofungin | beta t1/2 | = | 9 | hr | ALA5247142 | hr | ||||
2. | ALA1630575 | caspofungin | t1/2 | = | 8.1 | hr | ALA5247141 | hr | ||||
3. | ALA1630575 | caspofungin | CL | = | 0.21 | ml/min.kg | ALA5247140 | mL.min-1.kg-1 | ||||
4. | ALA1630575 | caspofungin | t1/2 | = | 5.2 | hr | ALA5247139 | hr | ||||
5. | ALA1630575 | caspofungin | CL | = | 0.26 | ml/min.kg | ALA5247138 | mL.min-1.kg-1 | ||||
6. | ALA1630575 | caspofungin | MFC | = | 0.125 | mg/ml | ALA5247137 | mg/ml | Candida albicans | |||
7. | ALA1630575 | caspofungin | IC50 | = | 0.6 | nM | ALA5247136 | 9.22 | nM | Candida albicans | ||
8. | ALA1630575 | caspofungin | IC50 | = | 6 | uM | ALA5128690 | 5.22 | nM | Homo sapiens | ||
9. | ALA1630575 | caspofungin | Activity | 0 | ALA5118925 | Active | ||||||
10. | ALA1630575 | caspofungin | Activity | 0 | ALA5118924 | Active | ||||||
11. | ALA1630575 | caspofungin | MIC80 | = | 0.016 | ug ml-1 | ALA5118851 | ug.mL-1 | Candida albicans | |||
12. | ALA1630575 | caspofungin | MIC80 | = | 0.125 | ug ml-1 | ALA5118850 | ug.mL-1 | Candida albicans | |||
13. | ALA1630575 | caspofungin | Activity | 0 | ALA5118807 | Active | ||||||
14. | ALA1630575 | caspofungin | Activity | 0 | ALA5118806 | Active | ||||||
15. | ALA1630575 | caspofungin | Activity | 0 | ALA5118805 | Active | ||||||
16. | ALA1630575 | caspofungin | MIC | > | 31.3 | ug ml-1 | ALA4413265 | ug.mL-1 | Aspergillus terreus | |||
17. | ALA1630575 | caspofungin | MIC | > | 31.3 | ug ml-1 | ALA4413264 | ug.mL-1 | Aspergillus nidulans | |||
18. | ALA1630575 | caspofungin | MIC | > | 31.3 | ug ml-1 | ALA4413263 | ug.mL-1 | Aspergillus flavus | |||
19. | ALA1630575 | caspofungin | MIC | = | 1.95 | ug ml-1 | ALA4413262 | ug.mL-1 | Candida parapsilosis | |||
20. | ALA1630575 | caspofungin | MIC | = | 0.48 | ug ml-1 | ALA4413261 | ug.mL-1 | Pichia kudriavzevii |