| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1630715 | 4m-(S) | IC50 | = | 400 | nM | ALA3887190 | 6.40 | 321168 | nM | Homo sapiens | |
| 2. | ALA1630715 | 4m-(S) | IC50 | = | 30 | nM | ALA3705247 | 7.52 | 213356 | nM | Homo sapiens | |
| 3. | ALA1630715 | 4m-(S) | IC50 | = | 170 | nM | ALA3707991 | 6.77 | 213373 | nM | Rattus norvegicus | |
| 4. | ALA1630715 | 4m-(S) | IC50 | = | 190 | nM | ALA3707969 | 6.72 | 213372 | nM | Homo sapiens | |
| 5. | ALA1630715 | 4m-(S) | Activity | 0 | ALA1640943 | Active | Rattus norvegicus | |||||
| 6. | ALA1630715 | 4m-(S) | Activity | 0 | ALA1640942 | Active | Rattus norvegicus | |||||
| 7. | ALA1630715 | 4m-(S) | Ratio | = | 6 | ALA1640941 | ||||||
| 8. | ALA1630715 | 4m-(S) | F | = | 98 | % | ALA1640940 | % | Rattus norvegicus | |||
| 9. | ALA1630715 | 4m-(S) | t1/2 | = | 3 | hr | ALA1640939 | hr | Rattus norvegicus | |||
| 10. | ALA1630715 | 4m-(S) | t1/2 | = | 1.8 | hr | ALA1640938 | hr | Rattus norvegicus | |||
| 11. | ALA1630715 | 4m-(S) | AUC | = | 120 | micromol.hr/L | ALA1640937 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 12. | ALA1630715 | 4m-(S) | AUC | = | 19 | micromol.hr/L | ALA1640936 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 13. | ALA1630715 | 4m-(S) | Drug uptake | = | 7.59 | umol/L | ALA1640935 | umol/L | Rattus norvegicus | |||
| 14. | ALA1630715 | 4m-(S) | Drug uptake | = | 1.59 | umol/L | ALA1640887 | umol/L | Rattus norvegicus | |||
| 15. | ALA1630715 | 4m-(S) | Tmax | = | 2 | hr | ALA1640886 | hr | Rattus norvegicus | |||
| 16. | ALA1630715 | 4m-(S) | Tmax | = | 2 | hr | ALA1640885 | hr | Rattus norvegicus | |||
| 17. | ALA1630715 | 4m-(S) | Cmax | = | 21.8 | umol/L | ALA1640884 | nM | Rattus norvegicus | |||
| 18. | ALA1630715 | 4m-(S) | Cmax | = | 3.5 | umol/L | ALA1640883 | nM | Rattus norvegicus | |||
| 19. | ALA1630715 | 4m-(S) | Vd | = | 2.6 | L/Kg | ALA1640882 | L.kg-1 | Rattus norvegicus | |||
| 20. | ALA1630715 | 4m-(S) | CL | = | 1.6 | L/hr/kg | ALA1640881 | mL.min-1.kg-1 | Rattus norvegicus |
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