| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1671936 | 28 | solubility | = | 1 | ug ml-1 | ALA3406919 | ug.mL-1 | ||||
| 2. | ALA1671936 | 28 | Ratio Ki | > | 1000 | ALA1679420 | ||||||
| 3. | ALA1671936 | 28 | Ratio Ki | = | 69 | ALA1679414 | ||||||
| 4. | ALA1671936 | 28 | Ratio Ki | = | 45 | ALA1679419 | ||||||
| 5. | ALA1671936 | 28 | Ki | > | 10000 | nM | ALA1679417 | nM | Homo sapiens | |||
| 6. | ALA1671936 | 28 | Tmax | = | 0.5 | hr | ALA1679430 | hr | Rattus norvegicus | |||
| 7. | ALA1671936 | 28 | CL | = | 0.3 | L/hr/kg | ALA1679433 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA1671936 | 28 | F | = | 88 | % | ALA1679432 | % | Rattus norvegicus | |||
| 9. | ALA1671936 | 28 | t1/2 | = | 1.2 | hr | ALA1679435 | hr | Rattus norvegicus | |||
| 10. | ALA1671936 | 28 | Vdss | = | 1 | L/Kg | ALA1679434 | L.kg-1 | Rattus norvegicus | |||
| 11. | ALA1671936 | 28 | Ratio | = | 0.8 | ALA1679429 | ||||||
| 12. | ALA1671936 | 28 | t1/2 | = | 7.8 | hr | ALA1679436 | hr | Rattus norvegicus | |||
| 13. | ALA1671936 | 28 | Papp | = | 67 | 10'6cm/s | ALA1679425 | 10'6cm/s | Homo sapiens | |||
| 14. | ALA1671936 | 28 | Papp | = | 88 | 10'6cm/s | ALA1679424 | 10'6cm/s | Homo sapiens | |||
| 15. | ALA1671936 | 28 | Cmax | = | 878 | mg/ml | ALA1679431 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 16. | ALA1671936 | 28 | Activity | 0 | ALA1679437 | Dose-dependent effect | Mus musculus | |||||
| 17. | ALA1671936 | 28 | Activity | 0 | ALA1679438 | Dose-dependent effect | Mus musculus | |||||
| 18. | ALA1671936 | 28 | INH | = | 36 | % | ALA1679418 | % | Homo sapiens | |||
| 19. | ALA1671936 | 28 | PPB | = | 85 | % | ALA1679428 | % | Homo sapiens | |||
| 20. | ALA1671936 | 28 | PPB | = | 87 | % | ALA1679427 | % | Canis lupus familiaris |
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