# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1681830 | 3, NCTFA | IC50 | = | 0.67 | uM | ALA2423971 | 6.17 | nM | Oryctolagus cuniculus | ||
2. | ALA1681830 | 3, NCTFA | Activity | = | 66 | % | ALA2423970 | % | Oryctolagus cuniculus | |||
3. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423968 | Not Active | Oryctolagus cuniculus | |||||
4. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423972 | Active | Oryctolagus cuniculus | |||||
5. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423966 | Active | Oryctolagus cuniculus | |||||
6. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423967 | Active | Oryctolagus cuniculus | |||||
7. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423962 | Active | ||||||
8. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423761 | Not Active | ||||||
9. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA2423758 | Active | ||||||
10. | ALA1681830 | 3, NCTFA | K | = | 5.74 | /s | ALA2423755 | /s | ||||
11. | ALA1681830 | 3, NCTFA | t1/2 | = | 121 | ms | ALA2423754 | hr | ||||
12. | ALA1681830 | 3, NCTFA | INH | = | 42 | % | ALA2423753 | % | Oryctolagus cuniculus | |||
13. | ALA1681830 | 3, NCTFA | INH | 0 | ALA2423971 | Dose-dependent effect | % | Oryctolagus cuniculus | ||||
14. | ALA1681830 | 3, NCTFA | Ratio EC50 | = | 10 | ALA1687482 | ||||||
15. | ALA1681830 | 3, NCTFA | Ratio EC50 | = | 10 | ALA1687481 | ||||||
16. | ALA1681830 | 3, NCTFA | EC50 | = | 0.88 | uM | ALA1687480 | 6.06 | nM | |||
17. | ALA1681830 | 3, NCTFA | EC50 | = | 0.88 | uM | ALA1687479 | 6.06 | nM | |||
18. | ALA1681830 | 3, NCTFA | INH | 0 | ALA1687477 | Active | % | Rattus norvegicus | ||||
19. | ALA1681830 | 3, NCTFA | INH | 0 | ALA1687476 | Active | % | Rattus norvegicus | ||||
20. | ALA1681830 | 3, NCTFA | Activity | 0 | ALA1687473 | Active | Rattus norvegicus |