# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1681882 | 18j | CLint | 38 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | |||||
2. | ALA1681882 | 18j | CLint | 11 | microL/min/mg | ALA3301370 | mL.min-1.g-1 | |||||
3. | ALA1681882 | 18j | Solubility | 91.2 | uM | ALA3301364 | nM | |||||
4. | ALA1681882 | 18j | IC50 | = | 0.2 | nM | ALA3119548 | 9.70 | nM | Homo sapiens | ||
5. | ALA1681882 | 18j | IC50 | = | 1.6 | nM | ALA1687492 | 8.80 | nM | Rattus norvegicus | ||
6. | ALA1681882 | 18j | IC50 | = | 1.1 | nM | ALA1687491 | 8.96 | nM | Mus musculus | ||
7. | ALA1681882 | 18j | AUC | = | 950 | nM.hr | ALA1687483 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
8. | ALA1681882 | 18j | IC50 | = | 0.2 | nM | ALA1687494 | 9.70 | nM | Homo sapiens | ||
9. | ALA1681882 | 18j | AUC | = | 0.95 | uM.hr | ALA5257223 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
10. | ALA1681882 | 18j | pKi | = | 9.5 | ALA5257222 | 9.50 | nM | Homo sapiens |