| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1683074 | 19 | Ratio | = | 3 | ALA1786457 | ||||||
| 2. | ALA1683074 | 19 | CL | = | 33.8 | ml/min.kg | ALA1786456 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 3. | ALA1683074 | 19 | TI | = | 3860 | ALA1786455 | ||||||
| 4. | ALA1683074 | 19 | t1/2 | = | 3.9 | hr | ALA1786454 | hr | Rattus norvegicus | |||
| 5. | ALA1683074 | 19 | IC50 | = | 3.2 | nM | ALA1786261 | 8.49 | nM | Homo sapiens | ||
| 6. | ALA1683074 | 19 | CL | = | 9.3 | microL/min/mg | ALA1786162 | mL.min-1.g-1 | Homo sapiens | |||
| 7. | ALA1683074 | 19 | Fu | = | 29 | % | ALA1786161 | Homo sapiens | ||||
| 8. | ALA1683074 | 19 | IC50 | = | 1.7 | uM | ALA1786160 | 5.77 | nM | Homo sapiens | ||
| 9. | ALA1683074 | 19 | IC50 | = | 3.9 | nM | ALA1786159 | 8.41 | nM | Homo sapiens | ||
| 10. | ALA1683074 | 19 | IC50 | = | 3 | nM | ALA1786158 | 8.52 | nM | Homo sapiens | ||
| 11. | ALA1683074 | 19 | F | = | 57 | % | ALA1686167 | % | Macaca fascicularis | |||
| 12. | ALA1683074 | 19 | AUC | = | 5.3 | uM.hr | ALA1686166 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca fascicularis | ||
| 13. | ALA1683074 | 19 | t1/2 | = | 3 | hr | ALA1686165 | hr | Macaca fascicularis | |||
| 14. | ALA1683074 | 19 | Vdss | = | 6.2 | L/Kg | ALA1686164 | L.kg-1 | Macaca fascicularis | |||
| 15. | ALA1683074 | 19 | CL | = | 2.2 | L/hr/kg | ALA1686163 | mL.min-1.kg-1 | Macaca fascicularis | |||
| 16. | ALA1683074 | 19 | F | = | 84 | % | ALA1686162 | % | Rattus norvegicus | |||
| 17. | ALA1683074 | 19 | AUC | = | 3 | uM.hr | ALA1686161 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 18. | ALA1683074 | 19 | t1/2 | = | 5 | hr | ALA1686160 | hr | Rattus norvegicus | |||
| 19. | ALA1683074 | 19 | Vdss | = | 17 | L/Kg | ALA1686159 | L.kg-1 | Rattus norvegicus | |||
| 20. | ALA1683074 | 19 | CL | = | 3.8 | L/hr/kg | ALA1686158 | mL.min-1.kg-1 | Rattus norvegicus |
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