# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1683440 | 24c | F | = | 38 | % | ALA1686367 | % | Rattus norvegicus | |||
2. | ALA1683440 | 24c | t1/2 | = | 1.2 | hr | ALA1686366 | hr | Rattus norvegicus | |||
3. | ALA1683440 | 24c | Vdss | = | 6 | L/Kg | ALA1686365 | L.kg-1 | Rattus norvegicus | |||
4. | ALA1683440 | 24c | CL | = | 93 | ml/min.kg | ALA1686364 | mL.min-1.kg-1 | Rattus norvegicus | |||
5. | ALA1683440 | 24c | AUC | = | 840 | nM.hr | ALA1686363 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
6. | ALA1683440 | 24c | EC50 | = | 0.24 | uM | ALA1686362 | 6.62 | nM | Homo sapiens | ||
7. | ALA1683440 | 24c | Ratio IC50 | = | 3 | ALA1686361 | ||||||
8. | ALA1683440 | 24c | Ratio IC50 | = | 9 | ALA1686360 | ||||||
9. | ALA1683440 | 24c | IC50 | > | 7.9 | uM | ALA1686359 | nM | Homo sapiens | |||
10. | ALA1683440 | 24c | INH | = | -2 | % | ALA1686358 | % | Homo sapiens | |||
11. | ALA1683440 | 24c | INH | = | -9 | % | ALA1686357 | % | Homo sapiens | |||
12. | ALA1683440 | 24c | INH | = | -4 | % | ALA1686356 | % | Homo sapiens | |||
13. | ALA1683440 | 24c | INH | = | 15 | % | ALA1686355 | % | Homo sapiens | |||
14. | ALA1683440 | 24c | INH | = | 29 | % | ALA1686354 | % | Homo sapiens | |||
15. | ALA1683440 | 24c | INH | = | 26 | % | ALA1686353 | % | Homo sapiens | |||
16. | ALA1683440 | 24c | INH | = | 37 | % | ALA1686352 | % | Homo sapiens | |||
17. | ALA1683440 | 24c | INH | = | 22 | % | ALA1686351 | % | Homo sapiens | |||
18. | ALA1683440 | 24c | INH | = | -2 | % | ALA1686350 | % | Rattus norvegicus | |||
19. | ALA1683440 | 24c | INH | = | 0 | % | ALA1686349 | % | Homo sapiens | |||
20. | ALA1683440 | 24c | INH | = | 85 | % | ALA1686348 | % | Homo sapiens |