# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1688558 | NSC-84094 | IC50 | = | 31.64 | uM | ALA4822994 | 4.50 | nM | Homo sapiens | ||
2. | ALA1688558 | NSC-84094 | Potency | 10 | uM | ALA3215270 | inconclusive | nM | ||||
3. | ALA1688558 | NSC-84094 | IC50 | = | 1.5 | uM | ALA4001885 | 5.82 | nM | Clostridium botulinum | ||
4. | ALA1688558 | NSC-84094 | Activity | = | 10 | uM | ALA4001886 | uM | Clostridium botulinum | |||
5. | ALA1688558 | NSC-84094 | Potency | 11.22 | uM | ALA3215017 | active | nM | ||||
6. | ALA1688558 | NSC-84094 | IC50 | = | 2.2 | uM | ALA3117199 | 5.66 | nM | Clostridium botulinum | ||
7. | ALA1688558 | NSC-84094 | Drug metabolism | = | 0.186 | uM/min.mg | ALA3117197 | uM/min.mg | Homo sapiens | |||
8. | ALA1688558 | NSC-84094 | t1/2 | = | 29.6 | min | ALA3117196 | hr | Homo sapiens | |||
9. | ALA1688558 | NSC-84094 | t1/2 | = | 11.4 | hr | ALA3117194 | hr | Homo sapiens | |||
10. | ALA1688558 | NSC-84094 | Stability | = | 78.7 | % | ALA3117195 | % | Homo sapiens | |||
11. | ALA1688558 | NSC-84094 | Drug metabolism | = | 0.637 | uM/min.mg | ALA3117193 | uM/min.mg | Rattus norvegicus | |||
12. | ALA1688558 | NSC-84094 | t1/2 | = | 8.6 | min | ALA3117192 | hr | Rattus norvegicus | |||
13. | ALA1688558 | NSC-84094 | t1/2 | = | 13.5 | hr | ALA3117191 | hr | Rattus norvegicus | |||
14. | ALA1688558 | NSC-84094 | Stability | = | 67.3 | % | ALA3117190 | % | Rattus norvegicus | |||
15. | ALA1688558 | NSC-84094 | solubility | = | 78 | nM | ALA3117189 | nM | ||||
16. | ALA1688558 | NSC-84094 | solubility | = | 1174 | uM | ALA3117187 | nM | ||||
17. | ALA1688558 | NSC-84094 | Potency | 3.548 | uM | ALA2354282 | inconclusive | nM | Homo sapiens | |||
18. | ALA1688558 | NSC-84094 | Potency | 35.481 | uM | ALA2354254 | inconclusive | nM | Homo sapiens | |||
19. | ALA1688558 | NSC-84094 | log GI50 (M) | -5.244 | ALA1963976 | inactive | nM | Homo sapiens | ||||
20. | ALA1688558 | NSC-84094 | log GI50 (M) | -5.908 | ALA1963981 | inactive | nM | Homo sapiens |