# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA71917 | T-98475 | Solubility | 38 | uM | ALA3301364 | nM | |||||
2. | ALA71917 | T-98475 | LogD7.4 | 3.5 | ALA3301363 | |||||||
3. | ALA71917 | T-98475 | Ki | = | 0.1 | nM | ALA4263113 | 10.00 | nM | Homo sapiens | ||
4. | ALA71917 | T-98475 | Ki | = | 0.2 | nM | ALA4263116 | 9.70 | nM | Homo sapiens | ||
5. | ALA71917 | T-98475 | pIC50 | = | 8.3 | ALA4263113 | 8.30 | nM | Homo sapiens | |||
6. | ALA71917 | T-98475 | Potency | 15.849 | uM | ALA3215169 | active | nM | ||||
7. | ALA71917 | T-98475 | Potency | 2.512 | uM | ALA3214913 | active | nM | ||||
8. | ALA71917 | T-98475 | IC50 | = | 60 | nM | ALA956660 | 7.22 | nM | Rattus norvegicus | ||
9. | ALA71917 | T-98475 | IC50 | = | 4 | nM | ALA956659 | 8.40 | nM | Macaca mulatta | ||
10. | ALA71917 | T-98475 | IC50 | = | 0.2 | nM | ALA956658 | 9.70 | nM | Homo sapiens | ||
11. | ALA71917 | T-98475 | Potency | = | 7.08 | um | ALA1614257 | 5.15 | Inconclusive | nM | Homo sapiens | |
12. | ALA71917 | T-98475 | IC50 | = | 0.2 | nM | ALA871108 | 9.70 | nM | Homo sapiens | ||
13. | ALA71917 | T-98475 | IC50 | = | 2 | nM | ALA871110 | 8.70 | nM | Homo sapiens | ||
14. | ALA71917 | T-98475 | IC50 | = | 60 | nM | ALA871111 | 7.22 | nM | Rattus norvegicus | ||
15. | ALA71917 | T-98475 | IC50 | = | 4 | nM | ALA871112 | 8.40 | nM | Homo sapiens | ||
16. | ALA71917 | T-98475 | IC50 | = | 0.6 | nM | ALA871113 | 9.22 | nM | Homo sapiens | ||
17. | ALA71917 | T-98475 | IC50 | 0 | ALA871114 | Not Determined | Homo sapiens | |||||
18. | ALA71917 | T-98475 | IC50 | = | 60 | nM | ALA831379 | 7.22 | nM | Rattus norvegicus | ||
19. | ALA71917 | T-98475 | IC50 | = | 60 | nM | ALA829515 | 7.22 | nM | Homo sapiens | ||
20. | ALA71917 | T-98475 | Ki | = | 60 | nM | ALA680268 | 7.22 | nM | Rattus norvegicus |