# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1760809 | 45 | IC50 | > | 4000 | nM | ALA1764829 | nM | Mus musculus | |||
2. | ALA1760809 | 45 | IC50 | > | 4000 | nM | ALA1764828 | nM | Homo sapiens | |||
3. | ALA1760809 | 45 | IC50 | = | 25 | uM | ALA1764827 | 4.60 | nM | Homo sapiens | ||
4. | ALA1760809 | 45 | IC50 | = | 26 | uM | ALA1764826 | 4.58 | nM | Homo sapiens | ||
5. | ALA1760809 | 45 | IC50 | = | 36 | uM | ALA1764825 | 4.44 | nM | Homo sapiens | ||
6. | ALA1760809 | 45 | F | = | 96 | % | ALA1764824 | % | Mus musculus | |||
7. | ALA1760809 | 45 | AUC | = | 7.6 | uM.hr.Kg/mg | ALA1764759 | uM.hr.Kg/mg | Mus musculus | |||
8. | ALA1760809 | 45 | t1/2 | = | 6.8 | hr | ALA1764823 | hr | Mus musculus | |||
9. | ALA1760809 | 45 | CL | = | 5 | ml/min.kg | ALA1764760 | mL.min-1.kg-1 | Mus musculus | |||
10. | ALA1760809 | 45 | Activity | = | 23 | % | ALA1764755 | % | Homo sapiens | |||
11. | ALA1760809 | 45 | EC50 | > | 30 | uM | ALA1764754 | nM | Homo sapiens | |||
12. | ALA1760809 | 45 | INH | = | 80 | % | ALA1764758 | % | Mus musculus | |||
13. | ALA1760809 | 45 | INH | = | 95 | % | ALA1764753 | % | Mus musculus | |||
14. | ALA1760809 | 45 | IC50 | = | 2.3 | nM | ALA1764757 | 8.64 | nM | Mus musculus | ||
15. | ALA1760809 | 45 | IC50 | = | 5.5 | nM | ALA1764756 | 8.26 | nM | Homo sapiens |