# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1761554 | 3 | IC50 | = | 0.09 | uM | ALA3395897 | 7.05 | nM | Homo sapiens | ||
2. | ALA1761554 | 3 | IC50 | = | 0.05 | uM | ALA3395896 | 7.30 | nM | Homo sapiens | ||
3. | ALA1761554 | 3 | IC50 | = | 0.31 | uM | ALA3395902 | 6.51 | nM | Rattus norvegicus | ||
4. | ALA1761554 | 3 | F | = | 28 | % | ALA1763402 | % | Rattus norvegicus | |||
5. | ALA1761554 | 3 | Cmax | = | 0.7 | uM | ALA1763401 | nM | Rattus norvegicus | |||
6. | ALA1761554 | 3 | AUC | = | 6.3 | uM.hr | ALA1763400 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
7. | ALA1761554 | 3 | Vd | = | 0.8 | l | ALA1763399 | l | Rattus norvegicus | |||
8. | ALA1761554 | 3 | t1/2 | = | 3 | hr | ALA1763398 | hr | Rattus norvegicus | |||
9. | ALA1761554 | 3 | CL | = | 3 | ml/min.kg | ALA1763397 | mL.min-1.kg-1 | Rattus norvegicus | |||
10. | ALA1761554 | 3 | Drug uptake | = | 7.17 | uM | ALA1763395 | uM | Mus musculus | |||
11. | ALA1761554 | 3 | Drug uptake | = | 17.8 | uM | ALA1763394 | uM | Mus musculus | |||
12. | ALA1761554 | 3 | IC50 | = | 0.31 | uM | ALA1763333 | 6.51 | nM | Homo sapiens | ||
13. | ALA1761554 | 3 | IC50 | = | 0.05 | uM | ALA1763332 | 7.30 | nM | Homo sapiens | ||
14. | ALA1761554 | 3 | IC50 | = | 0.09 | uM | ALA1763331 | 7.05 | nM | Homo sapiens |