| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1762530 | 12 | Solubility | 195 | uM | ALA3301364 | nM | |||||
| 2. | ALA1762530 | 12 | PPB | 91.82 | % | ALA3301365 | % | |||||
| 3. | ALA1762530 | 12 | LogD7.4 | 2.94 | ALA3301363 | |||||||
| 4. | ALA1762530 | 12 | CLint | 31.62 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | |||||
| 5. | ALA1762530 | 12 | Cmax | = | 17 | uM | ALA1763693 | nM | Mus musculus | |||
| 6. | ALA1762530 | 12 | AUC | = | 155 | uM.hr | ALA1763692 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 7. | ALA1762530 | 12 | Cmax | = | 15 | uM | ALA1763691 | nM | Mus musculus | |||
| 8. | ALA1762530 | 12 | AUC | = | 63 | uM.hr | ALA1763690 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 9. | ALA1762530 | 12 | INH | > | 10 | uM | ALA1763689 | uM | Homo sapiens | |||
| 10. | ALA1762530 | 12 | INH | > | 10 | uM | ALA1763688 | uM | Homo sapiens | |||
| 11. | ALA1762530 | 12 | INH | > | 10 | uM | ALA1763687 | uM | Homo sapiens | |||
| 12. | ALA1762530 | 12 | INH | > | 10 | uM | ALA1763686 | uM | Homo sapiens | |||
| 13. | ALA1762530 | 12 | INH | = | 7 | uM | ALA1763685 | uM | Homo sapiens | |||
| 14. | ALA1762530 | 12 | INH | 0 | ALA1763684 | Not Active | % | Homo sapiens | ||||
| 15. | ALA1762530 | 12 | INH | 0 | ALA1763683 | Not Active | % | Homo sapiens | ||||
| 16. | ALA1762530 | 12 | INH | 0 | ALA1763682 | Not Active | % | Homo sapiens | ||||
| 17. | ALA1762530 | 12 | INH | 0 | ALA1763681 | Not Active | % | Homo sapiens | ||||
| 18. | ALA1762530 | 12 | TDI | = | 50 | % | ALA1763680 | % | Homo sapiens | |||
| 19. | ALA1762530 | 12 | IC50 | = | 0.01 | uM | ALA1763679 | 8.00 | nM | Mus musculus | ||
| 20. | ALA1762530 | 12 | IC50 | = | 0.08 | uM | ALA1763678 | 7.10 | nM | Homo sapiens |
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